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DARAPLADIB

SynDRA canonical compound SYN0000011 — structure-anchored drug synonym record

All known targets

• PLA2G7
• PLA2G1B

Mechanisms of action (all sources)

• Phospholipase inhibitor
• PLA2G7 INHIBITOR
• LDL-associated phospholipase A2 inhibitor
• PLA2G1B MODULATOR

Drug classes

• Phospholipase A2 Inhibitors

Cross-references

• PubChem CID: 9939609
• ChEMBL: CHEMBL204021
• DrugBank: DB06311
• KEGG: D03650
• PDB: 5HV
• Wikipedia: Darapladib
• TTD: D0L5UO
• LINCS BRD: BRD-K19085898

Synonyms

• SB-480848
• SB 480848
• Darapladib (USAN)
• Darapladib (SB-480848)
• N-(2-(Diethylamino)ethyl)-2-(2-((4-fluorobenzyl)thio)-4-oxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidin-1-yl)-N-((4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)methyl)acetamide
• UI1U1MYH09
• CHEMBL204021
• N-[2-(Diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4,5,6,7-tetrahydro-4-oxo-N-[[4'-(trifluoromethyl)[1,1'-biphenyl]-4-yl]methyl]-1H-cyclopentapyrimidine-1-acetamide
• 1H-Cyclopentapyrimidine-1-acetamide, N-(2-(diethylamino)ethyl)-2-(((4-fluorophenyl)methyl)thio)-4,5,6,7-tetrahydro-4-oxo-N-((4'-(trifluoromethyl)(1,1'-biphenyl)-4-yl)methyl)-
• N-[2-(Diethylamino)ethyl]-2-{2-[(4-Fluorobenzyl)sulfanyl]-4-Oxo-4,5,6,7-Tetrahydro-1h-Cyclopenta[d]pyrimidin-1-Yl}-N-{[4'-(Trifluoromethyl)biphenyl-4-Yl]methyl}acetamide
• Darapladib [USAN:INN]
• UNII-UI1U1MYH09
• SB480848
• DARAPLADIB [MI]
• DARAPLADIB [INN]
• DARAPLADIB [JAN]
• Darapladib (JAN/USAN)
• DARAPLADIB [USAN]
• DARAPLADIB [WHO-DD]
• Darapladib; SB-480848
• MLS006010424
• GTPL6696
• SCHEMBL2742709
• DTXSID70189073
• HMS3653B13
• HMS3744E13
• BCP04908
• EX-A2245
• ZINC3842798
• BDBM50125265
• FD5008
• MFCD18251452
• s7520
• AKOS025290042
• BCP9000585
• CCG-270349
• CS-1035
• DB06311