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AZELASTINE
SynDRA canonical compound SYN0001285 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | HRH1 |
|---|
| Mechanism of action | Histamine receptor antagonist |
|---|
| Indication | conjunctivitis |
|---|
| Disease area | ophthalmology |
|---|
All known targets
- HRH1
- ABCB1
- ADRA1A
- ADRA1B
- Adra1a
- CHRM1
- CYP2C19
- HRH3
- HTR2B
- HTR2C
- KCNH2
Mechanisms of action (all sources)
- Histamine receptor antagonist
- HRH1 ANTAGONIST
- Histamine H1 receptor antagonist
Drug classes
- Histamine H1 Receptor Antagonists
- Histamine-1 Receptor Antagonist
- Anti-Allergic Agents
- Anti-Asthmatic Agents
- Bronchodilator Agents
- Enzyme Inhibitors
- Histamine Agents
- Histamine Antagonists
- Histamine H1 Antagonists
- Histamine H1 Antagonists, Non-Sedating
- Lipoxygenase Inhibitors
- Neurotransmitter Agents
ATC classes
- R01A · DECONGESTANTS AND OTHER NASAL PREPARATIONS FOR TOPICAL USE
- R06A · ANTIHISTAMINES FOR SYSTEMIC USE
- S01G · DECONGESTANTS AND ANTIALLERGICS
Cross-references
Synonyms
- azelastine hydrochloride
- azelastine HCl
- Azelastina
- NSC-758971
- Azelastinum
- Optivar
- Astelin (TN)
- Astepro (TN)
- Azelastina [INN-Spanish]
- Azelastine (INN)
- Azelastine [INN:BAN]
- Azelastinum [INN-Latin]
- Optivar (TN)
- 4-((4-Chlorophenyl)methyl)-2-(hexahydro-1-methyl-1H-azepin-4-yl)-1(2H)-phthalazinone hydrochloride
- 4-((4-chlorophenyl)methyl)-2-(hexahydro-1-methyl-1H-azepin-4-yl)-1(2H)-phthalazinone HCl
- 4-(4-chlorobenzyl)-2-(1-methylazepan-4-yl)phthalazin-1(2H)-one
- 4-(p-Chlorobenzyl)-2-(hexahydro-1-methyl-1H-azepin-4-yl)-1-(2H)-phthalazinone
- 4-(p-chlorobenzyl)-2-(N-methylperhydroazepinyl-(4))-1-(2H)-phthalazinone
- 4-[(4-chlorophenyl)methyl]-2-(1-methylazepan-4-yl)phthalazin-1(2H)-one
- 4-[(4-chlorophenyl)methyl]-2-(1-methylazepan-4-yl)phthalazin-1-one
- NSC 758971
- ZQI909440X
- CHEBI:2950
- a-5610
- Vividrin akut Azelastin
- RefChem:54397
- DTXCID502638
- R01AC03
- R06AX19
- S01GX07
- Optilast
- AZELASTINE [INN]
- BRN 0900747
- rac-Azelastine
- UNII-ZQI909440X
- HSDB 7991
- (+-)-Azelastine
- AZELASTINE [MI]
Reported adverse events
- Epistaxis
- Somnolence
- Headache
- Fatigue
- Nausea
- Sneezing
- Dizziness
- Pharyngitis
- Rhinitis
- Sinusitis
- Weight
- Dysgeusia
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