← SynDRA
ORPHENADRINE
SynDRA canonical compound SYN0002461 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | CYP2B6 |
|---|
| Mechanism of action | acetylcholine receptor antagonist |
|---|
| Indication | muscle pain |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- SLC6A2
- SCN9A
- HRH1
- SCN5A
- SCN4A
- SCN10A
- SCN1A
- ADRA2A
- SCN11A
- HTR6
- Hrh1
- KCNH2
Mechanisms of action (all sources)
- HRH1 ANTAGONIST
- Histamine H1 receptor antagonist
- SLC6A2 INHIBITOR
- Norepinephrine transporter inhibitor
- SCN1A BLOCKER
- Sodium channel alpha subunit blocker
- SCN5A BLOCKER
- SCN4A BLOCKER
- SCN7A BLOCKER
- SCN2A BLOCKER
- SCN9A BLOCKER
- SCN3A BLOCKER
Drug classes
- Anti-Dyskinesia Agents
- Antiparkinson Agents
- Central Nervous System Agents
- Cholinergic Agents
- Cholinergic Antagonists
- Cytochrome P-450 CYP2B6 Inhibitors
- Cytochrome P-450 Enzyme Inhibitors
- Enzyme Inhibitors
- Metabolic Side Effects of Drugs and Substances
- Muscarinic Antagonists
- Muscle Relaxants, Central
- Neuromuscular Agents
ATC classes
- M03B · MUSCLE RELAXANTS, CENTRALLY ACTING AGENTS
- N04A · ANTICHOLINERGIC AGENTS
Cross-references
Synonyms
- disipal
- orphenadine
- orphenadrin
- orphenadrine citrate
- orphenadrine hydrochloride
- orphenadrine (chloride)
- orphenadrine HCl
- Orfenadrina
- Mefenamine
- Invagesic
- Mialgin
- Norgesic
- Orphenadrin
- Orphengesic
- Antiflex
- Biorphen
- Brocadisipal
- Brocasipal
- Disipal
- Lysantin
- Mephenamine
- Methyldiphenylhydramine
- Myolin
- Myotrol
- ORP
- Orfro
- Orphenadine
- Orphenadinum
- Orphenadrinum
- Orphenate
- Orphenedrine
- Norflex Orphenadrine Citrate
- Sodium Mefenamine
- WS 2434
- Banflex (TN)
- Biorphen (TN)
- Brocasipal (TN)
- Disipal (TN)
Look up ORPHENADRINE in the interactive SynDRA portal →