BUPIVACAINE

SynDRA canonical compound SYN0003709 — structure-anchored drug synonym record

Clinical phase	Launched
Approval status	Approved · Rx/OTC
Primary target(s)	KCNA5 \| SCN10A \| SCN9A
Mechanism of action	sodium channel blocker
Indication	caudal epidural block \| lumbar epidural block \| peripheral nerve block
Disease area	neurology/psychiatry

All known targets

KCNA5
SCN10A
SCN4A
SCN5A
CYP2D6
HTR3A
KCND3
KCNH2
KCNK3
Kcnd3
Kcnk3
Kcnk9

Mechanisms of action (all sources)

SCN4A BLOCKER
Sodium channel protein type IV alpha subunit blocker
KCNA5 MODULATOR
SCN5A PORE BLOCKER
sodium channel blocker
SCN10A MODULATOR

Drug classes

Anesthetics
Anesthetics, Local
Central Nervous System Agents
Central Nervous System Depressants
Peripheral Nervous System Agents
Sensory System Agents
Amide Local Anesthetic

ATC classes

N01B · ANESTHETICS, LOCAL

Cross-references

PubChem CID: 2474
ChEMBL: CHEMBL1098
DrugBank: DB00297
ChEBI: CHEBI:3215
KEGG: D07552
RxNorm: 1375412
Wikipedia: Bupivacaine
TTD: D0A0FL
LINCS BRD: BRD-A01636364

Synonyms

Look up BUPIVACAINE in the interactive SynDRA portal →