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ELETRIPTAN
SynDRA canonical compound SYN0008338 — structure-anchored drug synonym record
| Clinical phase | Launched |
| Approval status | Approved · Rx/OTC |
| Primary target(s) | HTR1A | HTR1B | HTR1D | HTR1E | HTR1F | HTR2B | HTR7 |
| Mechanism of action | serotonin receptor agonist |
| Indication | migraine headache |
| Disease area | neurology/psychiatry |
All known targets
- HTR1B
- HTR1D
- HTR1F
- HTR1A
- HTR1E
- HTR2B
- HTR7
Mechanisms of action (all sources)
- HTR1F AGONIST
- Serotonin 1f (5-HT1f) receptor agonist
- HTR1B AGONIST
- Serotonin 1b (5-HT1b) receptor agonist
- HTR1D AGONIST
- Serotonin 1d (5-HT1d) receptor agonist
- serotonin receptor agonist
- HTR1B MODULATOR
- HTR1D MODULATOR
Drug classes
- Neurotransmitter Agents
- Serotonin Agents
- Serotonin Receptor Agonists
- Serotonin 1b Receptor Agonists
- Serotonin 1d Receptor Agonists
- Serotonin-1b and Serotonin-1d Receptor Agonist
ATC classes
- N02C · ANTIMIGRAINE PREPARATIONS
Cross-references
Synonyms
- eletriptan hydrobromide
- UK 116044-04
- UK-116,044
- relpax
- UK-116,044-04 FREE BASE
- UK-116044
- UK-116044-04 FREE BASE
- Relpax
- Eletriptanum
- UK116044
- Eletriptan (INN)
- Eletriptan [INN:BAN]
- Relpax (TN)
- UK-116044-04
- (R)-3-[(1-Methyl-2-pyrrolidinyl)methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-Indole
- (R)-5-[2-(Benzenesulfonyl)ethyl]-3-[(N-methylpyrrolidin-2-yl)methyl]-1H-indole
- 3-(((R)-1-Methyl-2-pyrrolidinyl)methyl)-5-(2-(phenylsulfonyl)ethyl)indole
- 3-{[(2R)-1-methylpyrrolidin-2-yl]methyl}-5-[2-(phenylsulfonyl)ethyl]-1H-indole
- 5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole
- eletriptanum
- CHEBI:50922
- DTXCID7026861
- RefChem:57394
- N02CC06
- UK-166044
- UK-166,044
- NCGC00181130-01
- ELETRIPTAN [INN]
- CAS-143322-58-1
- UNII-22QOO9B8KI
- MFCD00943792
- Eletriptan, Free Base
- ELETRIPTAN [MI]
- ELETRIPTAN [VANDF]
- GTPL40
- ELETRIPTAN [WHO-DD]
- SCHEMBL26719
- orb1710738
Reported adverse events
- Asthenia
- Dizziness
- Dry mouth
- Dyspepsia
- Dysphagia
- Headache
- Nausea
- Somnolence
- Arrhythmia
- Flushing
- Hypersensitivity
- Serotonin syndrome
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