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GSK-424887
SynDRA canonical compound SYN0039543 — structure-anchored drug synonym record
| Clinical phase | Phase 1 |
|---|
| Primary target(s) | EDNRA |
|---|
| Mechanism of action | endothelin receptor antagonist |
|---|
All known targets
Mechanisms of action (all sources)
- endothelin receptor antagonist
- TACR1 ANTAGONIST
- EDNRA ANTAGONIST
Cross-references
Synonyms
- GSK424887
- FR139317
- D-Alanine, N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl-1-methyl-D-tryptophyl-3-(2-pyridinyl)-
- FR 139317
- CHEMBL352396
- 2-((1-(Hexahydro-1H-azepinyl)carbonyl)amino-4-methylpentanoyl)-3-(-(1-methyl-1H-indolyl)propionyl)amino-3-(2-pyridyl)propionic acid
- D-Alanine, N-(N-(N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl)-1-methyl-D-tryptophyl)-3-(2-pyridinyl)-
- IYI99KCF2T
- RefChem:144527
- SCHEMBL29790472
- NS00073408
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