← SynDRA

INCB-057643

SynDRA canonical compound SYN0040039 — structure-anchored drug synonym record

All known targets

• BRD2
• BRD3
• BRD4

Mechanisms of action (all sources)

• BET bromodomain inhibitor

Drug classes

• Antineoplastic Agents

Cross-references

• PubChem CID: 118467751
• ChEMBL: CHEMBL4594412
• DrugBank: DB16054
• TTD: D7FJQ3

Synonyms

• INCB057643
• INCB 057643
• UNII-87TZD0JEBS
• 87TZD0JEBS
• 2,2,4-trimethyl-8-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-6-(methylsulfonyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
• 2,2,4-Trimethyl-8-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo(2,3-C)pyridin-4-yl)-6-(methylsulfonyl)-2H-benzo(b)(1,4)oxazin-3(4H)-one
• CHEMBL4594412
• SCHEMBL17200525
• US9957268, Example 75
• BDBM391587
• BCP29506
• EX-A1908
• NSC807398
• s8714
• NSC-807398
• BS-16298
• HY-111485
• AK00799038
• CS-0042192
• CC1(OC2=C(N(C1=O)C)C=C(C=C2C=2C1=C(C(N(C2)C)=O)NC=C1)S(=O)(=O)C)C
• 2,2,4-trimethyl-8-(6-methyl-7- oxo-6,7-dihydro-1H- pyrrolo[2,3-c]pyridin-4-yl)-6- (methylsulfonyl)-2H-1,4- benzoxazin-3(4H)-one
• 2H-1,4-Benzoxazin-3(4H)-one, 8-(6,7-dihydro-6-methyl-7-oxo-1H-pyrrolo(2,3-C)pyridin-4-yl)-2,2,4-trimethyl-6-(methylsulfonyl)-
• RefChem:148083
• BET Inhibitor INCB057643
• orb1301806
• SCHEMBL29422923
• INCB057643?
• INCB-057643?
• AKOS037515683
• AC-35555
• BI166425
• DA-64432
• PD132573
• SY389280
• T5417
• D80635